Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Sodium-dependent phosphate transporter 1 (Homo sapiens) | BDBM50341384 (CHEMBL4170023) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.50E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Inc. Curated by ChEMBL | Assay Description Inhibition of human Pit-1 expressed in HEK293 cells coexpressing tetracyclin assessed as reduction in uptake of 33P-radiolabeled Pi incubated for 20 ... | ACS Med Chem Lett 9: 440-445 (2018) Article DOI: 10.1021/acsmedchemlett.8b00013 BindingDB Entry DOI: 10.7270/Q26T0Q7K | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium-dependent phosphate transporter 1 (Homo sapiens) | BDBM50327362 (CHEMBL4159390) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 5.40E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Inc. Curated by ChEMBL | Assay Description Inhibition of human Pit-1 expressed in HEK293 cells coexpressing tetracyclin assessed as reduction in uptake of 33P-radiolabeled Pi incubated for 20 ... | ACS Med Chem Lett 9: 440-445 (2018) Article DOI: 10.1021/acsmedchemlett.8b00013 BindingDB Entry DOI: 10.7270/Q26T0Q7K | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium-dependent phosphate transporter 1 (Homo sapiens) | BDBM50327356 (CHEMBL4172584) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >1.40E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Inc. Curated by ChEMBL | Assay Description Inhibition of human Pit-1 expressed in HEK293 cells coexpressing tetracyclin assessed as reduction in uptake of 33P-radiolabeled Pi incubated for 20 ... | ACS Med Chem Lett 9: 440-445 (2018) Article DOI: 10.1021/acsmedchemlett.8b00013 BindingDB Entry DOI: 10.7270/Q26T0Q7K | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium-dependent phosphate transporter 1 (Homo sapiens) | BDBM50341383 (CHEMBL4175607) | UniProtKB/SwissProt GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >2.40E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Inc. Curated by ChEMBL | Assay Description Inhibition of human Pit-1 expressed in HEK293 cells coexpressing tetracyclin assessed as reduction in uptake of 33P-radiolabeled Pi incubated for 20 ... | ACS Med Chem Lett 9: 440-445 (2018) Article DOI: 10.1021/acsmedchemlett.8b00013 BindingDB Entry DOI: 10.7270/Q26T0Q7K | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium-dependent phosphate transporter 1 (Homo sapiens) | BDBM50327357 (CHEMBL4164986) | UniProtKB/SwissProt GoogleScholar AffyNet | Purchase PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | >2.40E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Inc. Curated by ChEMBL | Assay Description Inhibition of human Pit-1 expressed in HEK293 cells coexpressing tetracyclin assessed as reduction in uptake of 33P-radiolabeled Pi incubated for 20 ... | ACS Med Chem Lett 9: 440-445 (2018) Article DOI: 10.1021/acsmedchemlett.8b00013 BindingDB Entry DOI: 10.7270/Q26T0Q7K | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium-dependent phosphate transporter 1 (Homo sapiens) | BDBM50327355 (CHEMBL4164691) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >2.50E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Inc. Curated by ChEMBL | Assay Description Inhibition of human Pit-1 expressed in HEK293 cells coexpressing tetracyclin assessed as reduction in uptake of 33P-radiolabeled Pi incubated for 20 ... | ACS Med Chem Lett 9: 440-445 (2018) Article DOI: 10.1021/acsmedchemlett.8b00013 BindingDB Entry DOI: 10.7270/Q26T0Q7K | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium-dependent phosphate transporter 1 (Homo sapiens) | BDBM50327358 (CHEMBL4168403) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >2.50E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Inc. Curated by ChEMBL | Assay Description Inhibition of human Pit-1 expressed in HEK293 cells coexpressing tetracyclin assessed as reduction in uptake of 33P-radiolabeled Pi incubated for 20 ... | ACS Med Chem Lett 9: 440-445 (2018) Article DOI: 10.1021/acsmedchemlett.8b00013 BindingDB Entry DOI: 10.7270/Q26T0Q7K | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium-dependent phosphate transporter 1 (Homo sapiens) | BDBM50327363 (CHEMBL4176684) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >2.50E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Inc. Curated by ChEMBL | Assay Description Inhibition of human Pit-1 expressed in HEK293 cells coexpressing tetracyclin assessed as reduction in uptake of 33P-radiolabeled Pi incubated for 20 ... | ACS Med Chem Lett 9: 440-445 (2018) Article DOI: 10.1021/acsmedchemlett.8b00013 BindingDB Entry DOI: 10.7270/Q26T0Q7K | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium-dependent phosphate transporter 1 (Homo sapiens) | BDBM50327359 (CHEMBL4160507) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | >2.50E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Inc. Curated by ChEMBL | Assay Description Inhibition of human Pit-1 expressed in HEK293 cells coexpressing tetracyclin assessed as reduction in uptake of 33P-radiolabeled Pi incubated for 20 ... | ACS Med Chem Lett 9: 440-445 (2018) Article DOI: 10.1021/acsmedchemlett.8b00013 BindingDB Entry DOI: 10.7270/Q26T0Q7K | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium-dependent phosphate transporter 1 (Homo sapiens) | BDBM50341385 (CHEMBL4161567) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >2.50E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Inc. Curated by ChEMBL | Assay Description Inhibition of human Pit-1 expressed in HEK293 cells coexpressing tetracyclin assessed as reduction in uptake of 33P-radiolabeled Pi incubated for 20 ... | ACS Med Chem Lett 9: 440-445 (2018) Article DOI: 10.1021/acsmedchemlett.8b00013 BindingDB Entry DOI: 10.7270/Q26T0Q7K | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium-dependent phosphate transporter 1 (Homo sapiens) | BDBM50327361 (CHEMBL4172179) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >2.50E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Inc. Curated by ChEMBL | Assay Description Inhibition of human Pit-1 expressed in HEK293 cells coexpressing tetracyclin assessed as reduction in uptake of 33P-radiolabeled Pi incubated for 20 ... | ACS Med Chem Lett 9: 440-445 (2018) Article DOI: 10.1021/acsmedchemlett.8b00013 BindingDB Entry DOI: 10.7270/Q26T0Q7K | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium-dependent phosphate transporter 1 (Homo sapiens) | BDBM50327360 (CHEMBL4168827) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >6.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Inc. Curated by ChEMBL | Assay Description Inhibition of human Pit-1 expressed in HEK293 cells coexpressing tetracyclin assessed as reduction in uptake of 33P-radiolabeled Pi incubated for 20 ... | ACS Med Chem Lett 9: 440-445 (2018) Article DOI: 10.1021/acsmedchemlett.8b00013 BindingDB Entry DOI: 10.7270/Q26T0Q7K | |||||||||||
More data for this Ligand-Target Pair |